Thera-SAbDab

PATECIBART

>   Structural Summary
TherapeuticPatecibart
TargetEDNRA
Heavy ChainQVTLKESGPTLVKPTQTLTLTCTFSGFSLTTSGLGVAWIRQPPGKALEWLAHIWSDGDTRYYPALKNRLTITKDTSKNQVVLTMTNMDPVDTATYYCAHMKDDSLYFDNWGQGTLVTVSS
Light ChainEIVLTQSPDFQSVTPKEKVTITCRASQNIGTSIHWYQQKPDQYPKLLIKYASKSISGVPSRFSGSGSGTDFTLTINSLEAEDAATYYCQHSYSFPWTFGQGTKVEIK
100% seqID Fv StructureNone
99% seqID Fv StructureNone
95-98% seqID Fv StructureNone
>   Metadata
FormatWhole mAb
IsotypeG4
Highest Clinical Trial (Feb '25)Phase-I
Estimated Status (Feb '25)Discontinued
Recorded Developmental Technology
INN Year Proposed2023
INN Year Recommended2023
Companies InvolvedGmax Biopharm
Conditions Approvedna
Conditions Activena
Conditions DiscontinuedPulmonary arterial hypertension
Notes

Schneider, C., Raybould, M.I.J., Deane, C.M. (2022) SAbDab in the Age of Biotherapeutics: Updates including SAbDab-Nano, the Nanobody Structure Tracker. Nucleic Acids Res. 50(D1):D1368-D1372 [link]

SAbDab paper: Dunbar, J., Krawczyk, K. et al (2014). Nucleic Acids Res. 42. D1140-D1146 [link]

Thera-SAbDab paper: Raybould, M.I.J., Marks, C. et al (2019). Nucleic Acids Res. gkz827 [link]

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